Richard F Labaudinière: search on Z-Library

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1

Synthesis of a 10 000 Member 1,5-Benzodiazepine-2-one Library by the Directed Sorting Method

Herpin, Timothy F., Van Kirk, Katy G., Salvino, Joseph M., Yu, Sheng Tang, Labaudinière, Richard F.

Journal:

Journal of Combinatorial Chemistry

Year:

2000

Language:

english

File:

PDF, 219 KB

english, 2000

2

The Discovery of Tadalafil: A Novel and Highly Selective PDE5 Inhibitor. 1: 5,6,11,11a-Tetrahydro-1 H -imidazo[1‘,5‘:1,6]pyrido[3,4- b ]indole-1,3(2 H )-dione Analogues

Daugan, Alain, Grondin, Pascal, Ruault, Cécile, Le Monnier de Gouville, Anne-Charlotte, Coste, Hervé, Kirilovsky, Jorge, Hyafil, François, Labaudinière, Richard

Journal:

Journal of Medicinal Chemistry

Year:

2003

Language:

english

File:

PDF, 131 KB

english, 2003

3

Parallel Synthesis of Aldehydes and Ketone Facilitated by a New Solid-Phase Weinreb Amide †

Salvino, Joseph M., Mervic, Miljenko, Mason, Helen J., Kiesow, Terence, Teager, David, Airey, John, Labaudiniere, Richard

Journal:

Journal of Organic Chemistry

Year:

1999

Language:

english

File:

PDF, 236 KB

english, 1999

4

Synthesis of a New Fluoro-Wang Resin for Solid-Phase Reaction Monitoring by 19 F NMR Spectroscopy

Salvino, Joseph M., Patel, Sharmila, Drew, Mark, Krowlikowski, Paul, Orton, Edward, Kumar, N. Vassant, Caulfield, Thomas, Labaudiniere, Richard

Journal:

Journal of Combinatorial Chemistry

Year:

2001

Language:

english

File:

PDF, 38 KB

english, 2001

5

Novel applications of convertible isonitriles for the synthesis of mono and bicyclic γ-lactams via a UDC strategy

Christopher Hulme, Liang Ma, Marie-Pierre Cherrier, Joseph J Romano, George Morton, Celine Duquenne, Joseph Salvino, Richard Labaudiniere

Journal:

Tetrahedron Letters

Year:

2000

Language:

english

File:

PDF, 178 KB

english, 2000

6

Analogues of Human Parathyroid Hormone (1–31)NH2: Further Evaluation of the Effect of Conformational Constraint on Biological Activity

Stephen M Condon, Shelley Darnbrough, Christopher J Burns, Mark A Bobko, Isabelle Morize, Joanne Uhl, Navinchandra U Jariwala, Kathleen Burke, Richard F Labaudiniere

Journal:

Bioorganic & Medicinal Chemistry

Year:

2002

Language:

english

File:

PDF, 124 KB

english, 2002

7

.omega.-[(4,6-Diphenyl-2-pyridyl)oxy]alkanoic acid derivatives: a new family of potent and orally active LTB4 antagonists

Labaudiniere, Richard, Dereu, Norbert, Cavy, Francoise, Guillet, Marie Christine, Marquis, Olivier, Terlain, Bernard

Journal:

Journal of Medicinal Chemistry

Year:

1992

Language:

english

File:

PDF, 1.25 MB

english, 1992

8

Novel applications of carbon dioxide/MeOH for the synthesis of hydantoins and cyclic ureas via the Ugi reaction

Christopher Hulme, Liang Ma, Joseph J Romano, George Morton, Sheng-Yuh Tang, Marie-Pierre Cherrier, Steve Choi, Joseph Salvino, Richard Labaudiniere

Journal:

Tetrahedron Letters

Year:

2000

Language:

english

File:

PDF, 213 KB

english, 2000

9

Synthesis of novel proline and ψ-lactam derivatives as non-peptide mimics of Somatostatin/Sandostatin®

Dominique Damour, Frédéric Herman, Richard Labaudinière, Guy Pantel, Marc Vuilhorgne, Serge Mignani

Journal:

Year:

1999

Language:

english

File:

PDF, 1.20 MB

english, 1999

10

Removal of Thioacetal Protecting Groups by Cerium (IV) Ammonium Nitrate - Hydrolysis of 1,3-Dithiannes

Cristau, Henri-Jean, Chabaud, Bernard, Labaudinière, Richard, Christol, Henri

Journal:

Synthetic Communications

Year:

1981

Language:

english

File:

PDF, 191 KB

english, 1981

11

Novel applications of resin bound α-amino acids for the synthesis of benzodiazepines (via Wang resin) and ketopiperazines (via hydroxymethyl resin)

Christopher Hulme, Liang Ma, N.Vasant Kumar, Paul H Krolikowski, Andrew C Allen, Richard Labaudiniere

Journal:

Tetrahedron Letters

Year:

2000

Language:

english

File:

PDF, 240 KB

english, 2000

12

ChemInform Abstract: Improved Procedure for the Solution Phase Preparation of 1,4-Benzodiazepine-2,5-dione Libraries via Armstrong′s Convertible Isonitrile and the Ugi Reaction.

Christopher Hulme, John Peng, Sheng-Yuh Tang, Christopher J. Burns, Isabelle Morize, Richard Labaudiniere

Journal:

Year:

1999

Language:

english

File:

PDF, 30 KB

english, 1999

13

New indole derivatives as potent and selective serotonin uptake inhibitors

Serge Mignani, Dominique Damour, Adam Doble, Richard Labaudinière, Jean-Luc Malleron, Odile Piot, Claude Gueremy

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1993

Language:

english

File:

PDF, 447 KB

english, 1993

14

.omega.-[(.omega.-Arylalkyl)aryl]alkanoic acids: a new class of specific LTA4 hydrolase inhibitors

Labaudiniere, Richard, Hilboll, Gerd, Leon-Lomeli, Alicia, Lautenschlaeger, Hans Heiner, Parnham, Michael, Kuhl, Peter, Dereu, Norbert

Journal:

Journal of Medicinal Chemistry

Year:

1992

Language:

english

File:

PDF, 1.90 MB

english, 1992

15

ChemInform Abstract: RPR′s Approach to High-Speed Parallel Synthesis for Lead Generation

Richard F. Labaudiniere

Journal:

Year:

1999

File:

PDF, 24 KB

1999

16

Quaternary substituted PDE IV inhibitors II: The synthesis and in vitro evaluation of a novel series of γ-lactams

Christopher Hulme, Kevin Moriarty, Fu-Chih Huang, Jonathon Mason, Dan McGarry, Richard Labaudiniere, John Souness, Stevan Djuric

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1998

Language:

english

File:

PDF, 305 KB

english, 1998

17

ChemInform Abstract: A Convenient Synthetic Route to Macrocyclic cis-3-Phenylproline Derivatives as Mimics of Sandostatin®.

Dominique Damour, Gilles Doerflinger, Guy Pantel, Richard Labaudiniere, Jean-Pierre Leconte, Serge Sable, Marc Vuilhorgne, Serge Mignani

Journal:

Year:

1999

File:

PDF, 36 KB

1999

18

The Discovery of Tadalafil: A Novel and Highly Selective PDE5 Inhibitor. 2: 2,3,6,7,12,12a-hexahydropyrazino[1‘,2‘:1,6]pyrido[3,4- b ]indole-1,4-dione Analogues

Daugan, Alain, Grondin, Pascal, Ruault, Cécile, Le Monnier de Gouville, Anne-Charlotte, Coste, Hervé, Linget, Jean Michel, Kirilovsky, Jorge, Hyafil, François, Labaudinière, Richard

Journal:

Journal of Medicinal Chemistry

Year:

2003

Language:

english

File:

PDF, 183 KB

english, 2003

19

Improved Procedure for the Solution Phase Preparation of 1,4-Benzodiazepine-2,5-dione Libraries via Armstrong's Convertible Isonitrile and the Ugi Reaction

Hulme, Christopher, Peng, John, Tang, Sheng-Yuh, Burns, Christopher J., Morize, Isabelle, Labaudiniere, Richard

Journal:

Journal of Organic Chemistry

Year:

1998

Language:

english

File:

PDF, 76 KB

english, 1998

20

New 4-Point Pharmacophore Method for Molecular Similarity and Diversity Applications: Overview of the Method and Applications, Including a Novel Approach to the Design of Combinatorial Libraries Containing Privileged Substructures

Mason, Jonathan S., Morize, Isabelle, Menard, Paul R., Cheney, Daniel L., Hulme, Christopher, Labaudiniere, Richard F.

Journal:

Journal of Medicinal Chemistry

Year:

1999

Language:

english

File:

PDF, 359 KB

english, 1999

21

A Convenient Synthetic Route To Macrocyclic cis -3-Phenylproline Derivatives as Mimics of Sandostatin®

Damour, Dominique, Doerflinger, Gilles, Pantel, Guy, Labaudinière, Richard, Leconte, Jean-Pierre, Sablé, Serge, Vuilhorgne, Marc, Mignani, Serge

Journal:

Year:

1999

Language:

english

File:

PDF, 91 KB

english, 1999

22

Novel solid-phase synthesis of 1,5-benzothiazepine-4-one derivatives

George C Morton, Joseph M Salvino, Richard F Labaudinière, Timothy F Herpin

Journal:

Tetrahedron Letters

Year:

2000

Language:

english

File:

PDF, 160 KB

english, 2000

23

Synthesis and diversity analysis of lead discovery piperazine-2-carboxamide libraries

Timothy F. Herpin, George C. Morton, Allison K. Dunn, Cedric Fillon, Paul R. Menard, Sheng Yu Tang, Joseph M. Salvino, Richard F. Labaudinière

Journal:

Molecular Diversity

Year:

1998

Language:

english

File:

PDF, 264 KB

english, 1998

24

Orally active indole N-oxide PDE4 inhibitors

Christopher Hulme, Rose Mathew, Kevin Moriarty, Bruce Miller, Mercy Ramanjulu, Paul Cox, John Souness, Ken M. Page, Joanne Uhl, Jeffrey Travis, Richard Labaudiniere, Fu-chih Huang, Stevan W. Djuric

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1998

Language:

english

File:

PDF, 357 KB

english, 1998

25

The synthesis and biological evaluation of a novel series of indole PDE4 inhibitors I

Christopher Hulme, Kevin Moriarty, Bruce Miller, Rose Mathew, Mercy Ramanjulu, Paul Cox, John Souness, Ken M. Page, Joanne Uhl, Jeffrey Travis, Fu-chih Huang, Richard Labaudiniere, Stevan W. Djuric

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1998

Language:

english

File:

PDF, 363 KB

english, 1998

26

RPR's approach to high-speed parallel synthesis for lead generation

Richard F. Labaudiniere

Journal:

Drug Discovery Today

Year:

1998

Language:

english

File:

PDF, 148 KB

english, 1998

27

Synthesis of a regioselectively hexadeuterated linoleic acid

Viala, Jacques, Labaudiniere, Richard

Journal:

Journal of Organic Chemistry

Year:

1993

Language:

english

File:

PDF, 439 KB

english, 1993

28

Mechanism of Action and Clinical Application of Tafamidis in Hereditary Transthyretin Amyloidosis

Coelho, Teresa, Merlini, Giampaolo, Bulawa, Christine E., Fleming, James A., Judge, Daniel P., Kelly, Jeffery W., Maurer, Mathew S., Planté-Bordeneuve, Violaine, Labaudinière, Richard, Mundayat, Rajiv

Journal:

Neurology and Therapy

Year:

2016

Language:

english

File:

PDF, 1.29 MB

english, 2016

29

Parallel Solid-Phase Synthesis of Peptidyl Michael Acceptors

Caulfield, Thomas J., Patel, Sharmila, Salvino, Joseph M., Liester, Lara, Labaudiniere, Richard

Journal:

Journal of Combinatorial Chemistry

Year:

2000

Language:

english

File:

PDF, 75 KB

english, 2000

30

Synthesis and Binding Affinities of Novel Spirocyclic Lactam Peptidomimetics of Somatostatin

Damour, Dominique, Barreau, Michel, Blanchard, Jean-Charles, Burgevin, Marie-Claude, Doble, Adam, Pantel, Guy, Labaudinière, Richard, Mignani, Serge

Journal:

Chemistry Letters

Year:

1998

File:

PDF, 156 KB

1998

31

.omega.-[(.omega.-Arylalkyl)thienyl]alkanoic acids: from specific LTA4 hydrolase inhibitors to LTB4 receptor antagonists

Labaudiniere, Richard, Hilboll, Gerd, Leon-Lomeli, Alicia, Terlain, Bernard, Cavy, Francoise, Parnham, Michael, Kuhl, Peter, Dereu, Norbert

Journal:

Journal of Medicinal Chemistry

Year:

1992

Language:

english

File:

PDF, 1.31 MB

english, 1992

32

.omega.-[(4-Phenyl-2-quinolyl)oxy]alkanoic acid derivatives: a new family of potent LTB4 antagonists

Labaudiniere, Richard, Hendel, Wolfram, Terlain, Bernard, Cavy, Francoise, Marquis, Olivier, Dereu, Norbert

Journal:

Journal of Medicinal Chemistry

Year:

1992

Language:

english

File:

PDF, 1.09 MB

english, 1992

33

Novel safety-catch linker and its application with a Ugi/De-BOC/Cyclization (UDC) strategy to access carboxylic acids, 1,4-benzodiazepines, diketopiperazines, ketopiperazines and dihydroquinoxalinones

Christopher Hulme, John Peng, George Morton, Joseph M. Salvino, Tim Herpin, Richard Labaudiniere

Journal:

Tetrahedron Letters

Year:

1998

Language:

english

File:

PDF, 235 KB

english, 1998

34

Solid-Phase Horner−Emmons Synthesis of Olefins

Salvino, Joseph M., Kiesow, Terence J., Darnbrough, Shelley, Labaudiniere, Richard

Journal:

Journal of Combinatorial Chemistry

Year:

1999

Language:

english

File:

PDF, 67 KB

english, 1999

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